BMRB

Biological Magnetic Resonance Data Bank


A Repository for Data from NMR Spectroscopy on Proteins, Peptides, Nucleic Acids, and other Biomolecules
Member of WWPDB

BMRB Entry 34337

Title: Pepducin UT-Pep2 a biased allosteric agonist of Urotensin-II receptor

Deposition date: 2018-12-15 Original release date: 2020-01-13

Authors: Carotenuto, A.; Hoang, T.; Nassour, H.; Martin, R.; Billard, E.; Myriam, L.; Novellino, E.; Tanny, J.; Fournier, A.; Hebert, T.; Chatenet, D.

Citation: Hoang, T.; Nassour, H.; Martin, R.; Billard, E.; Myriam, L.; Novellino, E.; Carotenuto, A.; Tanny, J.; Fournier, A.; Hebert, T.; Chatenet, D.. "Membrane-tethered peptides derived from intracellular loops 2 and 3 of the urotensin II receptor act as allosteric agonists promoting Gq/Gi activation, EGFR transactivation and fibroblast proliferation"  . ., .-..

Assembly members:
entity_1, polymer, 14 residues, 1456.692 Da.

Natural source:   Common Name: Human   Taxonomy ID: 9606   Superkingdom: Eukaryota   Kingdom: Metazoa   Genus/species: Homo sapiens

Experimental source:   Production method: chemical synthesis

Entity Sequences (FASTA):
entity_1: XRPLDTVQRPKGYX

Data sets:
Data typeCount
1H chemical shifts95

Additional metadata:

  • Assembly
  • Samples and Experiments
  • Software
  • Spectrometers
  • Hide all